I-Top 10 Biologic Drugs e-United States

Ezi Ziyobisi Ziyakushintsha Indlela Yokugula Izifo

I-Biologics yilezi ziyobisi ezenziwe ngama-molecule eziyinkimbinkimbi ezenziwe ngezilwanyana ezincinci, izityalo, okanye iiseli zezilwanyana. Zininzi zezinto eziphilayo ziveliswa nge -teknoloji ye-DNA. Ngamanye amaxesha kuthiwa yi-biopharmaceuticals okanye iziyobisi ze-biological.

Iingcali zezinto eziphilayo ziye zatshintshelwa unyango lwezifo ezininzi ezinzulu kunye nezifo ezingapheliyo kwaye zidibanise izidakamizwa ezincinci zedolokhi ngaphandle kweentengiso eziphezulu. I-rheumatoid arthritis, iintsholongwane ezithile, kunye nesifo sikashukela sinenani elikhulu kakhulu lokunonyango lwe-biologic. I-Biologics iyatshintsha indlela iindlela oogqirha abaphatha ngayo iziganeko eziqhelekileyo eziye zaphazamisa abantu iminyaka.

Generic Biologics

Ngelixa ezininzi iziyobisi zingumakhemikhali owenziwe kwezinye iikhemikhali, i-biologics iyabiza kakhulu ngenxa yenkqubo yokuvelisa. Ngenxa yeendleko zabo eziphezulu, kukho imfuno enkulu yeenguqulelo zemveli zeyeza ze-biologic, ngakumbi ezilishumi ezibhalwe ngezantsi. Iinkampani ezininzi zonyango zifuna ukulungelelanisa ilungelo lokuvelisa iinguqulelo zesiGrike. Nangona kunjalo, ngenxa yokuba kunzima ukuvelisa, kukho iingxaki malunga nokukwazi ukuvelisa i-generics ngokukhuselekileyo nangokuthembekileyo.

EziPhambili ze-Biologics

Izidakamizwa ezilishumi ezibhalwe ngezantsi zigqithise kakhulu kakhulu inkcazo yemali ye "blockbuster" esichaza isiza njengokuba ivelise ngaphezu kweebhiliyoni eziyi-1 ngonyaka.

Ngo-2015, i-biologics yaqala ukujongana nokuncintisana nama- biosimilars , okanye i-biogenerics, xa i-Rituximab yaveliswa yi-IDEC Pharmaceuticals phantsi kwe- IDEC-C2B8 . [1] I-patent yase-US ikhishwe ngo-1998 kwaye yaphelelwa yisikhathi ngo-2015. I-Humira yalahlekelwa ukukhuselwa kwelungelo lobunikazi ngo-2016 kwaye i-Remicade iya kulahlekelwa ukukhuselwa kwayo ngo-2018.

Amanani angezantsi angokugqibela okufumaneka kwimveliso nganye.

  • 01 Humira

    Isigulana esichasayo-Humira asiyena kuphela i-biologic ethengiswa kakhulu; bekuyiziyobisi ezithengisa kakhulu emhlabeni jikelele, kungakhathaliseki ukuba yintoni iklasi.

    Iimpawu: I- rheumatoid arthritis, i-psqueasis ye-plaque, isifo sika-Crohn, isifo sezilonda zesilonda, i-spondylitis engavumelaniyo; i-psoriatic arthritis, i-polyarticular i-idiopathic arthritis

    Umkhiqizi: AbbVie, i-Abbott Laboratories iyahlulwa

    Ukuthengiswa kwehlabathi jikelele ngo-2015: i-$ 14 billion

    Igama lesiGrike : Adalimumab

    Umhla wokuqalisa: 2002

  • 02 Khuphela

    I-Remicade yenziwe yi-Centocor Ortho Biotech, ngoku iJanssen Biotech, i-subsidiary yaseJohnson & Johnson.

    Iimpawu: I- rheumatoid arthritis, isifo sikaCrohn, isifo se-spondylitis eskylosing, i-psoriatic arthritis, i-psqueasis ye-plaque, i-ulcerative colitis

    Umenzi: Johnson & Johnson / Merck & Co.

    Ukuthengiswa kwehlabathi jikelele ngo-2015: i $ 5.78 billion

    Igama lesiGrike : i- Infliximab

    Umhla wokuqalisa: 1998

  • 03 Rituxan

    I-Rituxan (rituximab) yaphuhliswa yi-IDEC Pharmaceuticals phantsi kwe-IDEC-C2B8. I-Rituxan okwangoku ithengiswa kwi-United States yi-Biogen Idec kunye ne-Roche subsidiary Genentech.

    Isibonakaliso: I- non-Hodgkins lymphoma, i-lymphocytic leukemia engapheliyo, i-rheumatoid arthritis

    Umenzi: Roche

    Ukuthengiswa kwehlabathi jikelele ngo-2015: i-$ 7.32 yezigidigidi

    Igama lesiGrike : Rituximab

    Umhla wokuqalisa: 1997

  • 04 Enbrel

    I-Etanercept yasungulwa ngabaphandi base-Immunex. Namhlanje isichengiselwano sithengiswa kwiNyakatho yeMerika ngo-Amgen kunye nePfizer, yiTata i-Pharmaceuticals eJapan kunye ne-Wyeth kulo lonke ihlabathi.

    Inkcazo: I- rheumatoid arthritis, i-plaque psoriasis, i-psoriatic arthritis

    Umenzi: uPfizer / Amgen

    Ukuthengiswa kwehlabathi jikelele ngo-2016: iibhiliyoni ezingama-23

    Igama lesiGrike : I- Etanercept

    Umhla wokuqalisa: 1998

  • 05 Lantus

    I-Lantus yaqulunqwa kwiziko lophando lwe-biotechnology laseSanofi-Aventis eFrankfurt-Höchst, eJamani.

    Isibonakaliso: Isifo sikashukela

    Umenzi: Sanofi

    Ukuthengiswa kwehlabathi jikelele ngo-2015: i-$ 6.98 yezigidigidi

    Igama lesiGrike : I- insulin glargine [i-rNNA origin] injection

    Umhla wokuqalisa: 2000

  • 06 Avastin

    Xa kuqaliswe ngo-2004, i-Avastin yakwaGenentech yayiyinye yezilwanyana ezibiza kakhulu kwiimarike, ene-$ 4,400 yamanani nganye ngenyanga.

    Isibonakaliso: Ubisi, i-colorectal, iinjongo, engekho encinci- i-glioblastoma, i-ovarian cancers

    Umenzi: Roche

    Ukuthengiswa kwehlabathi jikelele ngo-2015: i-$ 6.95 yezigidigidi

    Igama lesiGrike : Bevacizumab

    Umhla wokuqalisa: 2004

  • 07 Herceptin

    I-Herceptin yaphuhliswa nguGenentech, njengesixhamli seRoche, kunye neYunivesithi yaseCalina-Los Angeles yaseJonsson.

    Umqondiso: I- HER2 + yomhlaza wesifuba

    Umenzi: Roche

    Ukuthengiswa kwehlabathi jikelele ngo-2015: i-$ 6.59 yezigidigidi

    Igama lesiGrike : i- Trastuzumab

    Umhla wokuqalisa: 1998

  • 08 Neulasta

    Isibonakaliso: I- Neutropenia enxulumene nomhlaza wekhemotherapy

    Umenzi: Amgen

    Ukuthengiswa kwehlabathi jikelele ngo-2016: i $ 4.6 billion

    Igama lesiGrike : Pegfilgrastim

    Umhla wokuqalisa: 2002

  • 09 Lucentis

    Uphuhliswe nguGenentech, ranibizumab, injectable, ithengiswa eUnited States nguGenentech kunye noNovotis ngaphandle kwe-US

    Isibonakaliso: Ukuchithwa kwe-macular ukudala

    Umenzi: Roche, Novartis

    Ukuthengiswa kwehlabathi jikelele ngo-2015: i-$ 4.2 billion

    Igama lesiGrike : Ranibizumab

    Umhla wokuqalisa: 2006

  • 10 Avonex

    I-Avonex ithengiswa eUnited States yi-Biogen Idec kunye no-Merck phantsi kwegama legama elithi Rebif.

    I-Gemany's Fraunhofer Institute ye-Interfacial Engineering kunye ne-Biotechnology IGB kunye neCinnaGen Inkampani yathintela i-Interferon beta-1a kwaye ukususela ngo-2006 isiza sithengiswe njengeCinnoVex, i-biosimilar, e-Iran.

    Isibonakaliso: I- Multiple sclerosis (MS)

    Umenzi : Biogen Idec

    Ukuthengiswa kwehlabathi jikelele ngo-2014: iibhiliyoni ezingama-3

    Igama lesiGrike : i- Interferon beta-1a

    Umhla wokuqalisa: 1996

  • Ukuthembisa i-biologics kwipayipi:

    Kukho imithi eninzi ye-biologic ekugqibeleni, kuquka neziyobisi ukunyanga i-melanoma nezinye i-cancer. I-Sanofi ne-Regeneronhave babambisana ukuze bahlakulele i-Alirocumab, i-antibody monoclonal yokunyanga i-hypercholesterolemia. UJanssen ufumene "ukuqhubela phambili" kwe-FDA ukutyunjwa kwezobugcisa ekuphuhliseni unyango lwalo lwe-myeloma, iDaratumumab, i-antibody monoclonal. U-Merck uye wathola ukutyunjwa kobugcisa be-FDA ye-MK-3475, i-antibody monoclonal, ejoliswe kwi-melanoma ephezulu kunye nezinye i-cancer.